CAS NO. |
Products Name |
312636-16-1 |
SKI II |
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SKI-II is a synthetic inhibitor of sphingosine kinase (SK) activity with IC50 of 78 μM for SK1 and 45 μM for SK2. |
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1642300-52-4 |
KPT-8602 |
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KPT-8602 is a second-generation exportin-1 inhibitor, shows similar in vitro potency compared with KPT-330. |
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1088991-73-4 |
MK6096 |
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MK-6096(Filorexant) is an orally bioavailable potent and selective reversible antagonist of OX1 and OX2 receptor(<3 nM in binding). |
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110448-33-4 |
ML-7 hydrochloride |
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ML-7 Hcl is a cell-permeable, potent, reversible, ATP-competitive, and selective inhibitor of myosin light chain kinase (Ki = 300 nM); also inhibt smooth-muscle myosin light chain kinase, protein kinase C (PKC) and cAMP-dependent protein kinase (PKA). |
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794466-70-9 |
Vemakalant |
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Vernakalant(RSD-1235) is an investigational mixed ion channel blocker that can terminate acute atrial fibrillation (AF) in humans at 2 to 5 mg/kg and may be more atrial-selective than available agents; in treatment of antiarrhythmic. |
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266359-83-5 |
Repertaxin |
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Reparixin(DF 1681Y) is an inhibitor of CXCL8 receptor, also inhibit CXCR1 and CXCR2 activation, which has been shown to attenuate inflammatory responses in various injury models. |
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