CAS NO. |
Products Name |
223488-57-1 |
CP533536 |
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Evatanepag (CP-533536) is an EP2 receptor selective prostaglandin E2 (PGE2) agonist that induces local bone formation with EC50 of 0.3 nM. |
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866206-55-5 |
PRX08066 |
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PRX-08066 5-HT2B Maleic acid is a Selective Receptor Antagonist, IC50 for 3.4 nM, to act on rat model of MCT to prevent the severity of pulmonary hypertension. |
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1223403-58-4 |
LOXO-101 |
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LOXO-101 is a potent, ATP competitive TRK inhibitor with IC50s in low nanomolar range for inhibition of all TRK family members in binding and cellular assays, with 100x selectivity over other kinases, with 2 to 20 nM cellular potency against the TRKA, TRKB, and TRKC kinases. |
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869357-68-6 |
AZD8330 |
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AZD8330(ARRY-424704; ARRY-704) is a novel, selective, non-ATP competitive MEK 1/2 inhibitor with IC50 of 7 nM. |
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139180-30-6 |
ZM241385 |
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ZM 241385 is a novel non-xanthine adenosine receptor antagonist with selectivity for the A2a receptor subtype. |
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280744-09-4 |
SB216763 |
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SB 216763 is potent and selective glycogen synthase kinase-3 (GSK-3) inhibitor (Ki = 9 nM); competes with ATP. |
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403811-55-2 |
10058-F4 |
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10058-F4 is a cell-permeable thiazolidinone that specificallly inhibits the c-Myc-Max interaction and prevents transactivation of c-Myc target gene expression; induces cell-cycle arrest and apoptosis. |
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